SCHEMBL931601

SCHEMBL931601

COc1ccc(C2(C3CC3)N=C(C)C(N)=N2)cc1Br

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.50
KCNH2 Q12809 5/20 0.50
BACE2 Q9Y5Z0 2/20 0.47
APP P05067 7/20 0.37
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932191 0.82 BACE1 (0.51) BACE1KCNH2BACE2APP
SCHEMBL932236 0.77 BACE1 (0.53) BACE1KCNH2BACE2APPALDH1A1
SCHEMBL931716 0.74 BACE1 (0.78) BACE1KCNH2BACE2APP
SCHEMBL932205 0.73 BACE1 (0.61) BACE1KCNH2BACE2APP
SCHEMBL931327 0.73 BACE1 (0.53) BACE1KCNH2BACE2
SCHEMBL931861 0.73 BACE1 (0.53) BACE1KCNH2BACE2
SCHEMBL932399 0.73 BACE1 (0.53) BACE1KCNH2BACE2
SCHEMBL931281 0.72 BACE1 (0.60) BACE1KCNH2BACE2APP
SCHEMBL932626 0.71 BACE1 (0.65) BACE1KCNH2BACE2APP
SCHEMBL945923 0.71 ALDH1A1 (0.39) ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed