SCHEMBL931327

SCHEMBL931327

COc1ccc(C2(C3CCCCC3)N=C(C)C(N)=N2)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.53
KCNH2 Q12809 5/20 0.53
CYP3A4 P08684 1/20 0.46
CTSE P14091 1/20 0.46
CYP2C19 P33261 1/20 0.46
BACE2 Q9Y5Z0 1/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931861 1.00 BACE1 (0.53) BACE1KCNH2CYP3A4CTSECYP2C19
SCHEMBL932399 1.00 BACE1 (0.53) BACE1KCNH2CYP3A4CTSECYP2C19
SCHEMBL932679 0.76 BACE1 (0.41) BACE1KCNH2CYP3A4CTSECYP2C19
SCHEMBL932626 0.74 BACE1 (0.65) BACE1KCNH2BACE2
SCHEMBL931601 0.73 BACE1 (0.50) BACE1KCNH2BACE2
SCHEMBL931425 0.72 BACE1 (0.52) BACE1KCNH2BACE2
SCHEMBL931135 0.72 BACE1 (0.52) BACE1KCNH2BACE2
SCHEMBL931281 0.69 BACE1 (0.60) BACE1KCNH2BACE2
SCHEMBL931835 0.69 BACE1 (1.00) BACE1KCNH2CTSEBACE2
SCHEMBL945139 0.68 BACE1 (0.42) BACE1CYP3A4CTSECYP2C19SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed