SCHEMBL932236

SCHEMBL932236

COc1ccc(C2(C3CC3)N=C(C)C(N)=N2)cc1-c1cnccn1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.53
KCNH2 Q12809 6/20 0.47
BACE2 Q9Y5Z0 3/20 0.45
APP P05067 3/20 0.36
KLK3 P07288 1/20 0.34
CHEK1 O14757 1/20 0.34
CTSD P07339 1/20 0.33
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
HPGD P15428 1/20 0.32
NR4A1 P22736 1/20 0.32
ESR2 Q92731 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931611 0.85 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL931716 0.82 BACE1 (0.78) BACE1KCNH2BACE2APPCTSD
SCHEMBL931601 0.77 BACE1 (0.50) BACE1KCNH2BACE2APPALDH1A1
SCHEMBL932038 0.69 BACE1 (1.00) BACE1KCNH2BACE2APPCTSD
SCHEMBL14951105 0.69 KDM4E (0.48) KLK3CHEK1ALDH1A1POLBHPGD
SCHEMBL1075789 0.67 BACE1 (0.74) BACE1KCNH2BACE2APP
SCHEMBL931151 0.67 BACE1 (0.51) BACE1KCNH2BACE2ALDH1A1POLB
SCHEMBL931695 0.67 BACE1 (0.70) BACE1KCNH2BACE2APP
SCHEMBL931135 0.67 BACE1 (0.52) BACE1KCNH2BACE2APPCTSD
SCHEMBL931425 0.67 BACE1 (0.52) BACE1KCNH2BACE2APPHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed