SCHEMBL931802

SCHEMBL931802

CSC1=NC(c2cccc(Br)c2)(C2CCNCC2)N=C1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.38
KCNH2 Q12809 4/20 0.38
BACE2 Q9Y5Z0 2/20 0.38
CTSD P07339 1/20 0.33
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
SLC6A4 P31645 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CHRND Q07001 1/20 0.32
EP300 Q09472 1/20 0.30
HTR1A P08908 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945501 0.89 BACE1 (0.47) BACE1KCNH2BACE2CTSDHTR1A
SCHEMBL946218 0.87 BACE1 (0.49) BACE1KCNH2BACE2CTSDCHRNA1
SCHEMBL932745 0.84 BACE1 (0.37) BACE1KCNH2BACE2CTSD
SCHEMBL932230 0.76 BACE1 (0.59) BACE1KCNH2BACE2
SCHEMBL931281 0.74 BACE1 (0.60) BACE1KCNH2BACE2CTSD
SCHEMBL932626 0.73 BACE1 (0.65) BACE1KCNH2BACE2CTSD
SCHEMBL931210 0.71 BACE1 (0.47) BACE1KCNH2BACE2CTSDHTR1A
SCHEMBL931852 0.69 BACE1 (0.49) BACE1KCNH2BACE2CTSDCHRNA1
SCHEMBL946784 0.69 BACE1 (0.76) BACE1KCNH2BACE2
SCHEMBL946602 0.68 BACE1 (0.57) BACE1KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed