SCHEMBL931852

SCHEMBL931852

NC1=NC(c2cccc(Br)c2)(C2CCOCC2)N=C1S

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.49
KCNH2 Q12809 4/20 0.49
CTSD P07339 1/20 0.37
BACE2 Q9Y5Z0 2/20 0.36
CHRNA1 P02708 1/20 0.30
CHRNG P07510 1/20 0.30
CHRNB1 P11230 1/20 0.30
CHRNB2 P17787 1/20 0.30
SLC6A2 P23975 1/20 0.30
CHRNB4 P30926 1/20 0.30
SLC6A4 P31645 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30
SLC6A3 Q01959 1/20 0.30
CHRND Q07001 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931210 0.88 BACE1 (0.47) BACE1KCNH2CTSDBACE2
SCHEMBL946218 0.82 BACE1 (0.49) BACE1KCNH2CTSDBACE2CHRNA1
SCHEMBL932141 0.80 BACE1 (0.45) BACE1KCNH2CTSDBACE2
SCHEMBL932230 0.76 BACE1 (0.59) BACE1KCNH2BACE2
SCHEMBL931281 0.73 BACE1 (0.60) BACE1KCNH2CTSDBACE2
SCHEMBL932626 0.72 BACE1 (0.65) BACE1KCNH2CTSDBACE2
SCHEMBL945501 0.70 BACE1 (0.47) BACE1KCNH2CTSDBACE2
SCHEMBL931802 0.69 BACE1 (0.38) BACE1KCNH2CTSDBACE2CHRNA1
SCHEMBL932676 0.68 MAPT (0.38) BACE1CTSDBACE2
SCHEMBL932274 0.67 BACE1 (0.43) BACE1KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed