SCHEMBL932745

SCHEMBL932745

CSC1=NC(c2cccc(Br)c2)(C2CCN(C(C)(C)C)CC2)N=C1N

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.37
KCNH2 Q12809 5/20 0.37
BACE2 Q9Y5Z0 2/20 0.37
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
OPRM1 P35372 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
CTSD P07339 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945501 0.85 BACE1 (0.47) BACE1KCNH2BACE2CTSD
SCHEMBL931802 0.84 BACE1 (0.38) BACE1KCNH2BACE2CTSD
SCHEMBL946218 0.83 BACE1 (0.49) BACE1KCNH2BACE2CTSD
SCHEMBL932230 0.72 BACE1 (0.59) BACE1KCNH2BACE2
SCHEMBL931281 0.70 BACE1 (0.60) BACE1KCNH2BACE2CTSD
SCHEMBL932073 0.69 BACE1 (0.59) BACE1KCNH2BACE2CTSD
SCHEMBL6891103 0.69 BACE1 (0.56) BACE1KCNH2BACE2CTSD
SCHEMBL932626 0.69 BACE1 (0.65) BACE1KCNH2BACE2CTSD
SCHEMBL932141 0.67 BACE1 (0.45) BACE1KCNH2BACE2CTSD
SCHEMBL931210 0.67 BACE1 (0.47) BACE1KCNH2BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed