SCHEMBL932141

SCHEMBL932141

NC1=NC(c2cccc(Br)c2)(C2CCN(C(=O)O)CC2)N=C1S

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.45
CTSD P07339 1/20 0.35
L3MBTL3 Q96JM7 5/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
L3MBTL4 Q8NA19 1/20 0.34
KCNH2 Q12809 4/20 0.33
MBTD1 Q05BQ5 3/20 0.33
BACE2 Q9Y5Z0 2/20 0.33
OPRD1 P41143 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
HSD11B1 P28845 1/20 0.32
MGLL Q99685 1/20 0.32
HCAR3 P49019 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932073 0.87 BACE1 (0.59) BACE1CTSDL3MBTL3L3MBTL1L3MBTL4
SCHEMBL931210 0.82 BACE1 (0.47) BACE1CTSDKCNH2BACE2
SCHEMBL931852 0.80 BACE1 (0.49) BACE1CTSDKCNH2BACE2
SCHEMBL6891103 0.74 BACE1 (0.56) BACE1CTSDKCNH2BACE2
SCHEMBL932230 0.70 BACE1 (0.59) BACE1KCNH2BACE2
SCHEMBL932637 0.70 BACE1 (0.86) BACE1KCNH2BACE2
SCHEMBL6894163 0.70 BACE1 (0.43) BACE1CTSDKCNH2BACE2
SCHEMBL931281 0.69 BACE1 (0.60) BACE1CTSDKCNH2BACE2
SCHEMBL932626 0.68 BACE1 (0.65) BACE1CTSDKCNH2BACE2
SCHEMBL23852239 0.68 ALDH1A1 (0.43) BACE1CTSDL3MBTL3L3MBTL1L3MBTL4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed