SCHEMBL9320106

SCHEMBL9320106

COc1cc(C=CNC=O)cc(OC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 8/20 0.61
CYP1B1 Q16678 8/20 0.61
NQO2 P16083 5/20 0.52
CYP1A2 P05177 5/20 0.52
ABL1 P00519 3/20 0.52
BCR P11274 3/20 0.52
TTR P02766 3/20 0.52
PTGS2 P35354 3/20 0.52
ALOX5 P09917 3/20 0.52
ESR1 P03372 2/20 0.52
ABCB1 P08183 2/20 0.52
CYP19A1 P11511 2/20 0.52
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
AHR P35869 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320099 1.00 CYP1A1 (0.61) CYP1A1CYP1B1NQO2CYP1A2ABL1
SCHEMBL9322786 0.82 RELA (0.59) CYP1A1CYP1B1NQO2CYP1A2CYP19A1
SCHEMBL9322769 0.82 RELA (0.59) CYP1A1CYP1B1NQO2CYP1A2CYP19A1
SCHEMBL49339 0.80 ALDH1A1 (0.57) CYP1A1CYP1B1NQO2CYP1A2ABL1
SCHEMBL6233317 0.80 ALDH1A1 (0.57) CYP1A1CYP1B1NQO2CYP1A2ABL1
SCHEMBL49338 0.80 ALDH1A1 (0.57) CYP1A1CYP1B1NQO2CYP1A2ABL1
SCHEMBL23209621 0.78 ALDH1A1 (0.56) CYP1A1CYP1B1NQO2CYP1A2ABL1
SCHEMBL9320689 0.78 MAPT (0.60) CYP1A1CYP1B1TTRCYP19A1TUBB4A
SCHEMBL9320697 0.78 MAPT (0.60) CYP1A1CYP1B1TTRCYP19A1TUBB4A
SCHEMBL1743365 0.78 CYP1A1 (1.00) CYP1A1CYP1B1NQO2CYP1A2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440887-B1 Improvement in the total synthesis of Erbstatin analogs ERBA CARLO SPA (IT) 1994-01-26 EP disclosed
US-5130472-A TOTAL SYNTHESIS OF ERBSTATIN ANALOGS FARMITALIA CARLO ERBA S.R.L. (IT) 1992-07-14 US disclosed
EP-0440887-A1 Improvement in the total synthesis of Erbstatin analogs FARMITALIA CARLO ERBA S.r.l. (IT) 1991-08-14 EP disclosed