SCHEMBL9320152

SCHEMBL9320152

COc1ccccc1C(O)C(N)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.58
KMT2A Q03164 2/20 0.49
POLB P06746 2/20 0.47
HTT P42858 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA12 O43570 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320155 0.87 ACHE (0.52) ACHEKMT2APOLBHTTNPSR1
SCHEMBL9320774 0.83 ACHE (0.58) ACHEKMT2APOLBHTTNPSR1
SCHEMBL7259231 0.81 CA1 (0.60) POLBHTTNPSR1L3MBTL1IDO1
SCHEMBL9320762 0.81 ACHE (0.56) ACHEKMT2APTGS1PTGS2CA1
SCHEMBL9320074 0.81 ADRA1A (0.68) ACHEKMT2AHTTCA1CA2
SCHEMBL12665837 0.80 KMT2A (0.53) ACHEKMT2APOLBHTTNPSR1
SCHEMBL8749509 0.80 KMT2A (0.53) ACHEKMT2APOLBHTTNPSR1
SCHEMBL30550438 0.80 KMT2A (0.53) ACHEKMT2APOLBHTTNPSR1
SCHEMBL3645158 0.80 KMT2A (0.53) ACHEKMT2APOLBHTTNPSR1
SCHEMBL22190012 0.80 IDO1 (0.49) ACHEKMT2APOLBHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440887-B1 Improvement in the total synthesis of Erbstatin analogs ERBA CARLO SPA (IT) 1994-01-26 EP disclosed
US-5130472-A TOTAL SYNTHESIS OF ERBSTATIN ANALOGS FARMITALIA CARLO ERBA S.R.L. (IT) 1992-07-14 US disclosed
EP-0440887-A1 Improvement in the total synthesis of Erbstatin analogs FARMITALIA CARLO ERBA S.r.l. (IT) 1991-08-14 EP disclosed