SCHEMBL932083

SCHEMBL932083

CC1=NC(c2ccccc2)(c2cc(C)c(OC(F)F)c(C)c2)N=C1N

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.50
BACE2 Q9Y5Z0 3/20 0.50
KCNH2 Q12809 2/20 0.44
CTSD P07339 2/20 0.42
REN P00797 1/20 0.36
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932175 0.87 BACE1 (0.51) BACE1BACE2KCNH2CTSDAPP
SCHEMBL931679 0.82 BACE1 (0.77) BACE1BACE2KCNH2
SCHEMBL932089 0.80 BACE1 (0.62) BACE1BACE2KCNH2
SCHEMBL932392 0.77 BACE1 (0.65) BACE1BACE2KCNH2
SCHEMBL932267 0.74 GAA (0.47) BACE1BACE2KCNH2
SCHEMBL6919957 0.74 BACE1 (0.40) BACE1BACE2KCNH2
SCHEMBL932844 0.73 BACE1 (0.50) BACE1BACE2KCNH2CTSDREN
SCHEMBL932204 0.71 BACE1 (0.67) BACE1BACE2KCNH2APP
SCHEMBL4554677 0.71 BACE1 (0.46) BACE1BACE2CTSDRENAPP
SCHEMBL4311809 0.70 BACE1 (0.77) BACE1BACE2CTSDRENAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed