SCHEMBL9322677

SCHEMBL9322677

CC(=O)Oc1cccc(/C=C/NC=O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.51
CYP3A4 P08684 2/20 0.50
LMNA P02545 2/20 0.50
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 3/20 0.48
POLB P06746 1/20 0.48
MAPK1 P28482 1/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.46
KDM4E B2RXH2 2/20 0.46
TP53 P04637 2/20 0.46
ACHE P22303 2/20 0.46
TTR P02766 1/20 0.46
IMPDH2 P12268 1/20 0.46
EGFR P00533 1/20 0.45
CYP19A1 P11511 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9322687 1.00 BCHE (0.51) BCHECYP3A4LMNAMEN1KMT2A
SCHEMBL9320697 0.84 MAPT (0.60) CYP3A4LMNAMEN1KMT2AMAPT
SCHEMBL9320689 0.84 MAPT (0.60) CYP3A4LMNAMEN1KMT2AMAPT
SCHEMBL9322769 0.81 RELA (0.59) BCHECYP19A1MAOB
SCHEMBL9320085 0.81 MAPT (0.60) CYP3A4LMNAMEN1KMT2AMAPT
SCHEMBL9320094 0.81 MAPT (0.60) CYP3A4LMNAMEN1KMT2AMAPT
SCHEMBL9322786 0.81 RELA (0.59) BCHECYP19A1MAOB
SCHEMBL23343707 0.81 CYP3A4 (0.56) BCHECYP3A4LMNAMEN1KMT2A
SCHEMBL716894 0.81 KMT2A (0.60) BCHECYP3A4LMNAMEN1KMT2A
SCHEMBL716895 0.81 KMT2A (0.60) BCHECYP3A4LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440887-B1 Improvement in the total synthesis of Erbstatin analogs ERBA CARLO SPA (IT) 1994-01-26 EP disclosed
US-5130472-A TOTAL SYNTHESIS OF ERBSTATIN ANALOGS FARMITALIA CARLO ERBA S.R.L. (IT) 1992-07-14 US disclosed
EP-0440887-A1 Improvement in the total synthesis of Erbstatin analogs FARMITALIA CARLO ERBA S.r.l. (IT) 1991-08-14 EP disclosed