SCHEMBL932320

SCHEMBL932320

Oc1c(-c2ccccc2)ccc(Cl)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
HDAC4 P56524 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
BACE1 P56817 1/20 0.44
ALOX5 P09917 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
BCL2L1 Q07817 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HNF4A P41235 1/20 0.42
CLCN2 P51788 1/20 0.41
ESR2 Q92731 2/20 0.41
CSNK2A1 P68400 2/20 0.40
ESR1 P03372 1/20 0.40
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL380375 0.84 CYP2A6 (0.50) CYP2A6HDAC4HDAC2HDAC8HDAC6
SCHEMBL1513823 0.83 CYP2A6 (0.48) CYP2A6HDAC4HDAC2HDAC8HDAC6
SCHEMBL28152739 0.83 BACE1 (0.50) CYP2A6HDAC4HDAC2HDAC8HDAC6
SCHEMBL27749305 0.81 CYP2A6 (0.46) CYP2A6HDAC4HDAC2HDAC8HDAC6
Methane SCHEMBL28112790 0.81 BACE1 (0.48) CYP2A6HDAC4HDAC2HDAC8HDAC6
SCHEMBL1696360 0.80 CYP2A6 (0.50) CYP2A6BACE1ALOX5ALDH1A1CLCN2
SCHEMBL29983843 0.79 AHR (0.60) CYP2A6BACE1ALOX5ALDH1A1CLCN2
SCHEMBL381602 0.79 AHR (0.60) CYP2A6BACE1ALOX5ALDH1A1CLCN2
SCHEMBL31434466 0.79 CYP2A6 (0.45) CYP2A6HDAC4HDAC2HDAC8HDAC6
SCHEMBL28545688 0.79 ESR2 (0.50) CYP2A6HDAC4HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
EP-1494995-B1 3-AMINOPHENOL DERIVATIVES SUBSTITUTED IN THE 2-POSITION, AND DYES CONTAINING THESE COMPOUNDS PROCTER & GAMBLE (US) 2010-09-22 EP claimed
WO-2019143110-A1 ORGANIC COMPOUND AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME 주식회사 두산 2019-07-25 WO disclosed
EP-1871759-A1 BENZODIOXANE AND BENZODIOXOLANE DERIVATIVES AND USES THEREOF Wyeth a Corporation of the State of Delaware (US) 2008-01-02 EP disclosed
WO-2006116158-A1 BENZODIOXANE AND BENZODIOXOLANE DERIVATIVES AND USES THEREOF WYETH (US) 2006-11-02 WO disclosed
US-20060241172-A1 Benzodioxane and benzodioxolane derivatives and uses thereof WYETH (US) 2006-10-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060241172-A1 Benzodioxane and benzodioxolane derivatives and uses thereof HTR2C, HTR1D, HTR1A CYP2A6 481/4885HDAC4 2133/4885HDAC2 2042/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.