SCHEMBL9324010

SCHEMBL9324010

O=C(O)c1nc(-c2ccccc2)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.44
ALDH1A1 P00352 1/20 0.43
KDM4E B2RXH2 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
PDE10A Q9Y233 1/20 0.42
LDHA P00338 1/20 0.42
KMO O15229 1/20 0.41
RAB9A P51151 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CTRC Q99895 1/20 0.40
DHODH Q02127 1/20 0.40
PIN1 Q13526 2/20 0.40
CYP1A2 P05177 2/20 0.40
MAPK1 P28482 1/20 0.40
CASP1 P29466 1/20 0.40
CYP2C19 P33261 1/20 0.40
PDGFRB P09619 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27662263 0.89 TP53 (0.41) TP53ALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL4243696 0.85 MAP2K3 (0.47) TP53ALDH1A1KDM4ERAB9AMEN1
SCHEMBL27515966 0.84 KMO (0.51) ALDH1A1KDM4ELMNAKMORAB9A
SCHEMBL10622534 0.84 ALDH1A1 (0.45) ALDH1A1KDM4ESMN1; SMN2LMNALDHA
SCHEMBL28794429 0.84 MCL1 (0.49) MCL1
SCHEMBL8822098 0.81 PDGFRB (0.38) TP53ALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL11177529 0.81 AKT1 (0.43) TP53ALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL259469 0.81 GAA (0.51) ALDH1A1KDM4ESMN1; SMN2KMT2ACYP1A2
SCHEMBL14736658 0.80 ADORA3 (0.40) ALDH1A1KDM4ERAB9AMEN1KMT2A
SCHEMBL21336547 0.78 MEN1 (0.38) ALDH1A1KDM4ELMNARAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3978069-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DT) 1976-08-31 US claimed
CN-1088062-C Certain 4 -aminomethyl -2 -substituted imidazole derivatives and 2 -aminomethyl -4 -substituted imidazole derivatives, new classes of dopamine receptor subtype specific ligands NEUROGEN CORP (US) 2002-07-24 CN disclosed
CN-1177349-A Certain 4 -aminomethyl -2 -substituted imidazole derivatives and 2 -aminomethyl -4 -substituted imidazole derivatives, new classes of dopamine receptor subtype specific ligands NEUROGEN CORP (US) 1998-03-25 CN disclosed
EP-0365030-B1 Imidazole compound and process for preparing the same ISHIHARA SANGYO KAISHA (JP) 1994-01-26 EP disclosed
US-5023336-A Fungicides, biocides ISHIHARA SANGYO KAISHA LTD. (JP) 1991-06-11 US disclosed
EP-0365030-A1 Imidazole compound and process for preparing the same ISHIHARA SANGYO KAISHA, Ltd. (JP) 1990-04-25 EP disclosed