Bromide

Bromide

SCHEMBL9325877

Br.C1=C(c2cccc3ccccc23)CCNC1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 1/20 0.53
HTR2C P28335 9/20 0.56
KDM4E B2RXH2 3/20 0.56
ALDH1A1 P00352 3/20 0.56
MAPT P10636 2/20 0.56
DRD2 P14416 1/20 0.56
ALOX15 P16050 1/20 0.56
HSD17B10 Q99714 1/20 0.56
KHK P50053 1/20 0.48
HTR6 P50406 7/20 0.47
HTR2A P28223 2/20 0.47
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
RAD52 P43351 1/20 0.47
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
PMP22 Q01453 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9310529 0.98 HTR2C (0.58) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL5138820 0.98 HTR2C (0.58) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL14085318 0.81 NISCH (0.41) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL6812900 0.80 HTR6 (0.56) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL9032554 0.80 HTR2C (0.58) HTR2CMAPTDRD2SIGMAR1HTR6
SCHEMBL19297061 0.80 HTR2C (0.53) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL6551566 0.77 HTR6 (0.62) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL7166811 0.76 SLC6A3 (0.44) KDM4EALDH1A1MAPTHSD17B10GAA
SCHEMBL7538898 0.74 HTR2C (0.66) HTR2CKDM4EALDH1A1MAPTDRD2
SCHEMBL1106949 0.74 HTR2C (0.61) HTR2CKDM4EALDH1A1MAPTDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292761-A Piperidine, tetrahydropyridine and pyrrolidine compounds ADIR ET COMPAGNIE (FR) 1994-03-08 US disclosed
US-5260317-A Hypotensive agents ADIR ET COMPAGNIE (FR) 1993-11-09 US disclosed
US-5250544-A Hypotensive agents ADIR ET COMPAGNIE (FR) 1993-10-05 US disclosed