SCHEMBL9327905

SCHEMBL9327905

CCCCN(c1ccccc1)N1C(=O)CCC1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CASP1 P29466 1/20 0.41
BRCA1 P38398 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TACR1 P25103 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
CHRM2 P08172 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
SLC6A2 P23975 1/20 0.39
ESR1 P03372 1/20 0.38
TP53 P04637 2/20 0.38
MAPT P10636 2/20 0.38
MC4R P32245 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
NPC1 O15118 1/20 0.37
JAK2 O60674 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9326729 0.82 ALDH1A1 (0.50) MEN1KMT2ASMN1; SMN2CASP1BRCA1
SCHEMBL29150713 0.72 TACR1 (0.40) MEN1KMT2ASMN1; SMN2CASP1BRCA1
SCHEMBL11416004 0.71 TACR1 (0.43) TACR1CHRM2CHRM1CHRM3MC4R
SCHEMBL107013 0.67 CNR2 (0.49) MEN1KMT2AHSD17B10TDP1ESR1
SCHEMBL157807 0.67 MEN1 (0.51) MEN1KMT2ASMN1; SMN2CASP1BRCA1
SCHEMBL2589900 0.67 MEN1 (0.51) MEN1KMT2ASMN1; SMN2CASP1BRCA1
SCHEMBL4565560 0.66 ALDH1A1 (0.41) SMN1; SMN2NPSR1RAB9AALDH1A1HTT
SCHEMBL4186050 0.66 BCHE (0.44) MEN1KMT2ATDP1CHRM2CHRM1
SCHEMBL29664813 0.66 KDM4E (0.35) KMT2ASMN1; SMN2MAPTALDH1A1GAA
SCHEMBL7416028 0.66 TACR1 (0.44) TACR1CHRM2CHRM1CHRM3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0257433-B1 Method for the preparation of quinoline-2,3-dicarboxylic acid AMERICAN CYANAMID CO (US) 1994-03-23 EP disclosed
US-4757146-A Method for the preparation of quinoline-2,3-dicarboxylic acid AMERICAN CYANAMID COMPANY (US) 1988-07-12 US disclosed
EP-0257433-A2 Method for the preparation of quinoline-2,3-dicarboxylic acid AMERICAN CYANAMID COMPANY (US) 1988-03-02 EP disclosed