SCHEMBL9328262

SCHEMBL9328262

Nc1nc(SCc2ccccc2)nc2nc(-c3ccco3)nn12

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 9/20 0.67
ADORA2B P29275 7/20 0.67
ADORA2A P29274 13/20 0.64
ADORA1 P30542 9/20 0.64
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
MAPK1 P28482 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9328920 0.90 ADORA2B (0.66) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL9327336 0.87 ADORA3 (0.69) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL7828518 0.83 ADORA3 (0.73) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9264847 0.81 ADORA3 (1.00) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL9428040 0.79 ADORA2A (0.69) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL6624396 0.79 ADORA2A (0.67) ADORA3ADORA2BADORA2AADORA1MAPK1
SCHEMBL7834626 0.78 ADORA2A (1.00) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL9427973 0.78 ADORA2A (0.72) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9326095 0.77 ADORA2A (0.80) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL9428127 0.77 ADORA2A (0.67) ADORA3ADORA2BADORA2AADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US claimed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP claimed
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed