SCHEMBL9329299

SCHEMBL9329299

NC(=O)c1ccccc1C(=O)NCBr

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
HTT P42858 1/20 0.46
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
MAPT P10636 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KMT2A Q03164 1/20 0.44
APEX1 P27695 1/20 0.44
METAP2 P50579 1/20 0.42
CTNNB1 P35222 1/20 0.42
BCAT2 O15382 1/20 0.41
TAAR1 Q96RJ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2080518 0.85 TSHR (0.51) TSHRHTTKDM4EALDH1A1HPGD
SCHEMBL6903284 0.84 TSHR (0.58) TSHRHTTKDM4EALDH1A1HPGD
SCHEMBL2129167 0.82 TSHR (0.47) TSHRHTTKDM4EALDH1A1HPGD
SCHEMBL30415135 0.82 HTT (0.57) TSHRHTTALDH1A1HPGDMAPT
SCHEMBL308733 0.82 HTT (0.57) TSHRHTTALDH1A1HPGDMAPT
SCHEMBL9343951 0.82 MAPT (0.47) KDM4EALDH1A1MAPTKMT2A
SCHEMBL2778140 0.81 HTT (0.56) TSHRHTTALDH1A1HPGDMAPT
SCHEMBL6566957 0.81 TSHR (0.55) TSHRHTTKDM4EALDH1A1HPGD
SCHEMBL6075765 0.81 TSHR (0.46) TSHRHTTKDM4EALDH1A1HPGD
SCHEMBL16486722 0.80 TSHR (0.54) TSHRHTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304549-A Control or prevention of degenerative joint diseases HOFFMANN-LA ROCHE INC. (US) 1994-04-19 US disclosed
EP-0497192-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-08-05 EP disclosed
US-4120688-A AMINOMETHYLPHOSPHONIC ACID THE PROCTOR & GAMBLE COMPANY (US) 1978-10-17 US disclosed