SCHEMBL9329574

SCHEMBL9329574

Nc1nc(NC2CCCCC2)nc2nc(-c3cccs3)nn12

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.64
ADORA3 P0DMS8 10/20 0.64
ADORA1 P30542 9/20 0.64
ADORA2B P29275 1/20 0.64
CSNK1D P48730 2/20 0.60
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 3/20 0.45
GAA P10253 3/20 0.45
GFER P55789 1/20 0.45
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9327282 0.78 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2BCSNK1D
SCHEMBL9326962 0.76 ADORA2A (0.98) ADORA2AADORA3ADORA1ADORA2BCSNK1D
SCHEMBL29117428 0.76 SMN1; SMN2 (0.46) KDM4EALDH1A1GAAGFERMAPT
SCHEMBL9327228 0.76 ADORA2A (0.67) ADORA2AADORA3ADORA1ADORA2BCSNK1D
SCHEMBL9327253 0.75 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2BCSNK1D
SCHEMBL9327337 0.75 ADORA2A (0.69) ADORA2AADORA3ADORA1ADORA2BCSNK1D
SCHEMBL7240698 0.71 KDM4E (0.49) KDM4EALDH1A1GAAGFERMAPT
SCHEMBL9328560 0.70 ADORA3 (0.58) ADORA2AADORA3ADORA1ADORA2BKDM4E
SCHEMBL30596777 0.69 KDM4E (0.41) ADORA2AADORA3ADORA1ADORA2BKDM4E
SCHEMBL30596780 0.69 KDM4E (0.41) ADORA2AADORA3ADORA1ADORA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed