SCHEMBL9328560

SCHEMBL9328560

CSc1nc(N)n2nc(-c3cccs3)nc2n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.58
ADORA2B P29275 2/20 0.58
LMNA P02545 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ADORA1 P30542 3/20 0.40
ADORA2A P29274 4/20 0.38
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
TP53 P04637 2/20 0.37
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9328936 0.85 ADORA3 (0.42) ADORA3ADORA2BLMNANPC1ADORA1
SCHEMBL23840696 0.78 ADORA3 (0.64) ADORA3ADORA2BLMNANPC1RAB9A
SCHEMBL30596777 0.75 KDM4E (0.41) ADORA3ADORA2BLMNANPC1ADORA1
SCHEMBL30596780 0.75 KDM4E (0.41) ADORA3ADORA2BLMNANPC1ADORA1
SCHEMBL9327253 0.74 ADORA2A (0.48) ADORA3ADORA2BADORA1ADORA2AALDH1A1
SCHEMBL9264847 0.74 ADORA3 (1.00) ADORA3ADORA2BADORA1ADORA2AKDM4E
SCHEMBL23291195 0.74 ADORA3 (0.58) ADORA3ADORA2BLMNANPC1RAB9A
SCHEMBL9327189 0.73 ADORA3 (0.61) ADORA3ADORA2BNPC1RAB9AADORA1
SCHEMBL7749219 0.73 ADORA3 (0.57) ADORA3ADORA2BLMNANPC1RAB9A
SCHEMBL9328272 0.72 ADORA3 (0.47) ADORA3ADORA2BNPC1RAB9AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed