SCHEMBL9329929

SCHEMBL9329929

O=C(NCCO[N+](=O)[O-])c1csc(-c2ccccc2[N+](=O)[O-])n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HPGDS O60760 1/20 0.43
PANK3 Q9H999 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
ACKR3 P25106 1/20 0.40
EIF4E P06730 5/20 0.40
DDX3X O00571 1/20 0.40
HIF1A Q16665 1/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC3 O15379 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9331226 0.88 PANK3 (0.47) CYP2C9CYP2C19HPGDSPANK3CYP1A2
SCHEMBL9329368 0.85 CYP2C9 (0.57) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9329277 0.80 HPGDS (0.46) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9328754 0.79 MEN1 (0.60) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9329461 0.78 MEN1 (0.48) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9328726 0.77 HIF1A (0.54) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9331727 0.77 MEN1 (0.50) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9329229 0.77 MEN1 (0.47) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL9329984 0.76 RAB9A (0.55) CYP2C9CYP2C19MEN1KMT2AALOX15
SCHEMBL6185761 0.76 ACHE (0.56) HPGDSEIF4EDDX3X

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300400-B1 Nitric acid ester derivative FUJISAWA PHARMACEUTICAL CO (JP) 1994-03-16 EP disclosed
US-5010093-A Vasodilators; cardiovascular disorders FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-04-23 US disclosed
US-4923886-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-05-08 US disclosed
EP-0300400-A1 Nitric acid ester derivative FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-01-25 EP disclosed