SCHEMBL9331128

SCHEMBL9331128

O=C(O)C(=NO)C(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 12/20 0.56
CES1 P23141 11/20 0.56
CYP2C19 P33261 2/20 0.47
GAA P10253 1/20 0.47
TSHR P16473 2/20 0.44
DAO P14920 1/20 0.44
NAPRT Q6XQN6 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
PARP1 P09874 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25324982 1.00 CES2 (0.56) CES2CES1CYP2C19GAATSHR
Methane SCHEMBL9572458 0.98 CES2 (0.54) CES2CES1CYP2C19GAATSHR
SCHEMBL1369324 0.91 CES2 (0.62) CES2CES1CYP2C19GAATSHR
SCHEMBL16597945 0.83 PARP10 (0.53) CES2CES1ALDH1A1POLBRAB9A
SCHEMBL16597944 0.83 PARP10 (0.53) CES2CES1ALDH1A1POLBRAB9A
SCHEMBL11416768 0.83 CES2 (0.61) CES2CES1CYP2C19GAATSHR
SCHEMBL1372210 0.83 CES2 (0.61) CES2CES1CYP2C19GAATSHR
SCHEMBL1370084 0.83 CES2 (0.61) CES2CES1CYP2C19GAATSHR
SCHEMBL7991738 0.81 NAPRT (0.50) CYP2C19GAANAPRTALDH1A1MAPT
SCHEMBL8913168 0.81 CES2 (0.58) CES2CES1MAPTL3MBTL1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114644634-A Pyrrole derivative and preparation method and application thereof 深圳市祥根生物医药有限公司 2022-06-21 CN disclosed
CN-107207470-B Antifungal agent F2G有限公司 2019-12-03 CN disclosed
CN-109982704-A Pharmaceutical preparation F2G有限公司 2019-07-05 CN disclosed
CN-107207470-A Antifungal agent F2G有限公司 2017-09-26 CN disclosed
EP-0220923-B1 Dipeptides and process GRACE W R & CO (US) 1994-04-27 EP disclosed
EP-0574028-A1 Dipeptide analogs of aspertame and process to prepare them as well as a new preparation of aspertame HAMPSHIRE CHEMICAL CORP. (US) 1993-12-15 EP disclosed
US-4873359-A Process for preparing as partyl-phenylalanine dipeptides W. R. GRACE & CO. - CONN. (US) 1989-10-10 US disclosed
US-4810817-A ARTIFICIAL SWEETENERS W. R. GRACE & CO. (US) 1989-03-07 US disclosed
US-4710583-A ENZYMATIC COUPLING OF PHENYLSERINE WITH ASPARTIC ACID; HYDROGENATION W. R. GRACE & CO. (US) 1987-12-01 US disclosed
EP-0220923-A2 Dipeptides and process W.R. Grace & Co.-Conn. (US) 1987-05-06 EP disclosed