SCHEMBL9331908

SCHEMBL9331908

CCNCC(C)N1c2ccccc2Sc2ccc(C#N)c(OC(=O)/C=C/C(=O)Oc3c(C#N)ccc4c3N(C(C)CNCC)c3ccccc3S4)c21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 9/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
TSHR P16473 1/20 0.35
MAPT P10636 3/20 0.34
GAA P10253 1/20 0.34
ACHE P22303 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HTT P42858 1/20 0.34
FNTA P49354 5/20 0.33
FNTB P49356 5/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
POLB P06746 1/20 0.32
ATM Q13315 1/20 0.32
HTR1A P08908 1/20 0.32
ADRB3 P13945 1/20 0.32
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9331918 0.74 BCHE (0.39) BCHECYP2D6CYP2C19TSHRMAPT
Fumaric Acid SCHEMBL9331904 0.74 BCHE (0.39) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9784933 0.72 BCHE (0.38) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9331357 0.71 LMNA (0.41) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9758897 0.71 LMNA (0.41) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9784853 0.71 BCHE (0.37) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9759527 0.70 PTGS1 (0.37) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9759522 0.70 PTGS1 (0.37) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9759380 0.69 BCHE (0.35) BCHECYP2D6CYP2C19TSHRMAPT
SCHEMBL9784916 0.69 BCHE (0.39) BCHECYP2D6CYP2C19TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5321026-A Antispasmodic agents RHONE-POULENC RORER S.A. (FR) 1994-06-14 US disclosed
US-5049669-A Also diuretics RHONE-POULENC SANTE (FR) 1991-09-17 US disclosed
US-4985419-A Analgesics, Diuretics RHONE-POULENC SANTE (FR) 1991-01-15 US disclosed