SCHEMBL9337098

SCHEMBL9337098

Cc1nc2cnccc2n1-c1ccc(COc2ccccc2C(=O)O)cc1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 1/20 0.43
HSD17B10 Q99714 1/20 0.42
DRD1 P21728 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523919 0.91 PARP1 (0.49) DRD1
SCHEMBL9335569 0.90 KMT2A (0.44)
SCHEMBL9386887 0.85 SGMS2 (0.58) SGMS2
SCHEMBL7770156 0.79 DRD1 (0.45) DRD1
Fumaric Acid SCHEMBL9868255 0.78 MEN1 (0.44) DRD1
Fumaric Acid SCHEMBL9868247 0.78 MEN1 (0.44) DRD1
SCHEMBL4446308 0.77 MRGPRX4 (0.58) HSD17B10
SCHEMBL9868989 0.77 MEN1 (0.42) HSD17B10
SCHEMBL9332773 0.76 MYC (0.50) HSD17B10
SCHEMBL7505146 0.75 HSD17B10 (0.59) HSD17B10DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533695-B1 IMIDAZO (4,5-c) PYRIDINES WITH PAF ANTAGONIST ACTIVITY PFIZER (US) 1994-10-05 EP disclosed
US-5322847-A Inhibit platelet activating factor, block leukotriene D4 receptors PFIZER INC. (US) 1994-06-21 US disclosed
EP-0533695-A1 IMIDAZO (4,5-c) PYRIDINES WITH PAF ANTAGONIST ACTIVITY. PFIZER (US) 1993-03-31 EP disclosed
EP-0530207-A1 IMIDAZOPYRIDINE PAF ANTAGONISTS Pfizer Limited (GB) 1993-03-10 EP disclosed
WO-1991017162-A1 IMIDAZOPYRIDINE PAF ANTAGONISTS PFIZER LIMITED (GB) 1991-11-14 WO disclosed
WO-1991017163-A1 IMIDAZO (4,5-c) PYRIDINES WITH PAF ANTAGONIST ACTIVITY PFIZER INC. (US) 1991-11-14 WO disclosed