SCHEMBL933900

SCHEMBL933900

NC(=O)CCCc1ccc(-c2ccncc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.51
MMP12 P39900 1/20 0.50
MMP13 P45452 1/20 0.50
CYP11B1 P15538 2/20 0.44
CYP21A2 P08686 1/20 0.44
CHUK O15111 1/20 0.44
HRH1 P35367 2/20 0.43
FFAR1 O14842 3/20 0.42
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP11B2 P19099 1/20 0.42
HDAC2 Q92769 1/20 0.41
TBK1 Q9UHD2 1/20 0.41
RARB P10826 1/20 0.41
TBXAS1 P24557 1/20 0.41
FAAH O00519 1/20 0.41
CES1 P23141 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1286084 0.89 HRH1 (0.53) CYP17A1HRH1FFAR1HDAC2TBXAS1
SCHEMBL10769953 0.83 HRH1 (0.57) CYP17A1HRH1FFAR1TBXAS1FAAH
SCHEMBL933474 0.82 PRKCI (0.57) CYP17A1CYP11B1CHUKROCK2CYP3A4
SCHEMBL6027 0.82 MKNK1 (0.58) TBXAS1
SCHEMBL31351850 0.81 HRH1 (0.60) HRH1HDAC2TBXAS1FAAHCES1
SCHEMBL11262500 0.81 FFAR1 (0.63) MMP12MMP13FFAR1HDAC2
SCHEMBL7369203 0.81 HRH1 (0.60) HRH1HDAC2TBXAS1FAAHCES1
SCHEMBL18248576 0.81 HRH1 (0.60) HRH1HDAC2TBXAS1FAAHCES1
SCHEMBL8813877 0.80 MAOB (0.53) FFAR1HDAC2
SCHEMBL28103661 0.79 CYP17A1 (0.56) CYP17A1MMP12MMP13CYP11B1CHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed