SCHEMBL9339077

SCHEMBL9339077

COC(=O)c1ccc(=O)n(CCNC(=O)c2ccc(C)nc2)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
ALDH1A1 P00352 2/20 0.48
CYP19A1 P11511 1/20 0.48
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GAA P10253 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
EPHX2 P34913 1/20 0.42
POLB P06746 2/20 0.41
ALOX15 P16050 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
CD274 Q9NZQ7 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9343034 0.88 MEN1 (0.52) KDM4EALDH1A1LMNAKMT2AGAA
SCHEMBL9339094 0.85 ALDH1A1 (0.52) ALDH1A1LMNAKMT2ATDP1POLB
SCHEMBL27380810 0.84 KDM4E (0.49) KDM4EALDH1A1CYP19A1KMT2ATDP1
SCHEMBL9343014 0.82 KMT2A (0.51) KDM4ELMNAKMT2AGAAEPHX2
SCHEMBL9339739 0.82 EPHX2 (0.54) KDM4EALDH1A1LMNAKMT2AGAA
SCHEMBL9339122 0.81 DRD2 (0.48) HDAC1ALOX15
SCHEMBL9341043 0.81 KMT2A (0.54) KDM4ELMNAKMT2APOLBALOX15
SCHEMBL9339176 0.80 KMT2A (0.54) KDM4EALDH1A1LMNAKMT2AGAA
SCHEMBL9339746 0.79 SMN1; SMN2 (0.53) ALDH1A1LMNAKMT2ATDP1EPHX2
SCHEMBL28887010 0.79 GAA (0.53) KDM4EALDH1A1LMNAKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360808-A Cardiovascular disorders, antispasmodic agents, hypotensive disorders, brains, anticonvulsants and antiepileptics HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-01 US disclosed
EP-0556738-A1 Pyridinylcarbonylaminoalkyl-dihydro-oxo-pyridines, their production and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-08-25 EP disclosed
CN-1075480-A New aryl carbonylamino alkyl-dihydro-oxo pyridine compounds and production thereof and application HOECHST AG (US) 1993-08-25 CN disclosed