SCHEMBL9339188

SCHEMBL9339188

O=C(O)c1ccc(=O)n(NC(=O)c2cccnc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
ALDH1A1 P00352 2/20 0.53
APP P05067 1/20 0.53
HCAR3 P49019 1/20 0.53
HCAR2 Q8TDS4 1/20 0.53
TSHR P16473 2/20 0.50
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PTGS2 P35354 2/20 0.47
LMNA P02545 2/20 0.46
THRB P10828 1/20 0.46
HIF1A Q16665 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP3A4 P08684 1/20 0.45
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339146 0.86 TSHR (0.61) ALDH1A1TSHRHDAC1HDAC6POLB
SCHEMBL27535821 0.79 TSHR (0.51) GAAALDH1A1TSHRHDAC1HDAC6
SCHEMBL9339116 0.76 SMN1; SMN2 (0.53) ALDH1A1TSHRTHRBMEN1KMT2A
SCHEMBL9341135 0.74 ALDH1A1 (0.58) ALDH1A1TSHRTHRBMEN1KMT2A
Niacin SCHEMBL30945735 0.74 ALDH1A1 (0.95) GAAALDH1A1APPHCAR3HCAR2
Niacin SCHEMBL29585450 0.74 ALDH1A1 (0.95) GAAALDH1A1APPHCAR3HCAR2
Niacin SCHEMBL1992336 0.74 ALDH1A1 (0.95) GAAALDH1A1APPHCAR3HCAR2
Niacin SCHEMBL4503958 0.74 ALDH1A1 (0.95) GAAALDH1A1APPHCAR3HCAR2
SCHEMBL30977158 0.73 ALDH1A1 (0.51) GAAALDH1A1APPHCAR3HCAR2
Niacin SCHEMBL29167280 0.72 ALDH1A1 (0.91) GAAALDH1A1APPHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360808-A Cardiovascular disorders, antispasmodic agents, hypotensive disorders, brains, anticonvulsants and antiepileptics HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-01 US disclosed
EP-0556738-A1 Pyridinylcarbonylaminoalkyl-dihydro-oxo-pyridines, their production and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-08-25 EP disclosed