SCHEMBL9339146

SCHEMBL9339146

COC(=O)c1ccc(=O)n(NC(=O)c2cccnc2)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.61
ALDH1A1 P00352 3/20 0.58
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HPGD P15428 1/20 0.46
KDM4E B2RXH2 2/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
USP2 O75604 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339188 0.86 GAA (0.53) TSHRALDH1A1MAPK1NPSR1HDAC1
SCHEMBL9339094 0.78 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1USP2LMNA
SCHEMBL9339746 0.76 SMN1; SMN2 (0.53) TSHRALDH1A1KMT2AMEN1LMNA
Methyl Nicotinate SCHEMBL29386553 0.76 ALDH1A1 (1.00) TSHRALDH1A1HPGDHDAC1HDAC6
Methyl Nicotinate SCHEMBL24566 0.76 ALDH1A1 (1.00) TSHRALDH1A1HPGDHDAC1HDAC6
Methyl Nicotinate SCHEMBL820747 0.76 ALDH1A1 (1.00) TSHRALDH1A1HPGDHDAC1HDAC6
Methyl Nicotinate SCHEMBL30779127 0.74 ALDH1A1 (0.96) TSHRALDH1A1HPGDHDAC1HDAC6
Methyl Nicotinate SCHEMBL29527047 0.74 ALDH1A1 (0.96) TSHRALDH1A1HPGDHDAC1HDAC6
Methyl Nicotinate SCHEMBL11491005 0.74 ALDH1A1 (0.96) TSHRALDH1A1HPGDHDAC1HDAC6
Methyl Nicotinate SCHEMBL28370871 0.74 ALDH1A1 (0.96) TSHRALDH1A1HPGDHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360808-A Cardiovascular disorders, antispasmodic agents, hypotensive disorders, brains, anticonvulsants and antiepileptics HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-01 US disclosed
EP-0556738-A1 Pyridinylcarbonylaminoalkyl-dihydro-oxo-pyridines, their production and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-08-25 EP disclosed
CN-1075480-A New aryl carbonylamino alkyl-dihydro-oxo pyridine compounds and production thereof and application HOECHST AG (US) 1993-08-25 CN disclosed