SCHEMBL9339796

SCHEMBL9339796

O=C(CN1CCC(COCc2ccccc2)CC1)c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.57
HTR2C P28335 1/20 0.57
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340596 0.94
Hydrochloric Acid SCHEMBL9341744 0.93
SCHEMBL7310558 0.80 DRD2 (0.67) HTR2AHTR2C
SCHEMBL10587379 0.79 ALDH1A1 (0.57) HTR2AHTR2CKCNH2
SCHEMBL7296727 0.78
SCHEMBL29208105 0.78 HTR2A (0.52) HTR2AHTR2CKCNH2
SCHEMBL9343644 0.77 HTR2A (0.59) HTR2AHTR2CKCNH2
SCHEMBL9341776 0.77 KDM4E (0.59)
SCHEMBL9339578 0.76 MEN1 (0.51) HTR2AHTR2CKCNH2
Hydrochloric Acid SCHEMBL9340630 0.76 HTR2A (0.58) HTR2AHTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0317997-B1 1,4-Disubstituted-piperidinyl compounds MERRELL DOW PHARMA (US) 1994-06-15 EP claimed
US-4870083-A 1,4-Disubstituted-piperidinyl compounds useful as analgesics and muscle relaxants MERRELL DOW PHARMACEUTICALS INC. (US) 1989-09-26 US claimed
CN-1034202-A 1, the 4-Disubstituted-piperidnyl compounds MERRELL DOW PHARMA (US) 1989-07-26 CN claimed
EP-0317997-A2 1,4-Disubstituted-piperidinyl compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1989-05-31 EP claimed
EP-0317997-B1 1,4-Disubstituted-piperidinyl compounds MERRELL DOW PHARMA (US) 1994-06-15 EP disclosed
US-4870083-A 1,4-Disubstituted-piperidinyl compounds useful as analgesics and muscle relaxants MERRELL DOW PHARMACEUTICALS INC. (US) 1989-09-26 US disclosed
CN-1034202-A 1, the 4-Disubstituted-piperidnyl compounds MERRELL DOW PHARMA (US) 1989-07-26 CN disclosed
EP-0317997-A2 1,4-Disubstituted-piperidinyl compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1989-05-31 EP disclosed