SCHEMBL9340840

SCHEMBL9340840

CC1(C)CC(O)(c2ccccn2)c2cc(Br)ccc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.42
ALDH1A1 P00352 1/20 0.38
PDK2 Q15119 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
ADRA1A P35348 1/20 0.35
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SLC11A2 P49281 1/20 0.33
SLC6A2 P23975 1/20 0.33
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PRMT5 O14744 2/20 0.32
WDR77 Q9BQA1 2/20 0.32
NR3C1 P04150 1/20 0.31
NLRP3 Q96P20 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340053 0.82 PDK2 (0.41) PDK2SLC11A2BACE1
SCHEMBL9340806 0.82 TP53 (0.37) TP53ALDH1A1PDK2ADRA1AMAPT
SCHEMBL9339974 0.79 ALDH1A1 (0.36) TP53ALDH1A1CA1CA2CA4
SCHEMBL9339933 0.79 TP53 (0.40) TP53ALDH1A1PDK2CA1CA2
SCHEMBL8311974 0.74 BACE1 (0.37) TP53ALDH1A1MAPTSLC6A2KMT2A
SCHEMBL8310390 0.71 SLC6A2 (0.36) TP53ALDH1A1SLC6A2NR3C1BACE1
SCHEMBL9340819 0.69 APP (0.40) TP53ALDH1A1PDK2TDP1L3MBTL1
SCHEMBL30725601 0.68 TP53 (0.62) TP53ALDH1A1ADRA1AMAPTL3MBTL1
SCHEMBL29143018 0.68 TP53 (0.62) TP53ALDH1A1ADRA1AMAPTL3MBTL1
SCHEMBL9344209 0.67 TP53 (0.36) TP53ALDH1A1PDK2ADRA1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356915-A Antihypertensive and bronchodilator agents J. URIACH & CIA. S.A. (ES) 1994-10-18 US disclosed
EP-0600147-A1 Tetralones with pharmacological activity, compositions containing them and process for their preparation J. URIACH & CIA. S.A. (ES) 1994-06-08 EP disclosed