SCHEMBL9340819

SCHEMBL9340819

OC1(c2ccccn2)CCCc2ccc(Br)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.40
BACE1 P56817 1/20 0.40
TP53 P04637 1/20 0.38
SIGMAR1 Q99720 1/20 0.36
KDM1A O60341 1/20 0.35
PDK2 Q15119 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
CYP17A1 P05093 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
AKR1B1 P15121 1/20 0.34
ALDH1A1 P00352 1/20 0.34
AVPR1A P37288 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339909 0.81 TRPV3 (0.41) SIGMAR1KDM1AGRIN1GRIN2AGRIN2B
SCHEMBL9341809 0.79 HSD11B1 (0.35) SIGMAR1PDK2GRIN1GRIN2AGRIN2B
SCHEMBL9339996 0.78 BACE1 (0.41) APPBACE1TP53SIGMAR1KDM1A
SCHEMBL9339933 0.78 TP53 (0.40) TP53PDK2GRIN1GRIN2AGRIN2B
SCHEMBL6902549 0.75 SIGMAR1 (0.43) SIGMAR1KDM1APDK2GRIN1GRIN2A
SCHEMBL8126674 0.74 CYP3A4 (0.47) SIGMAR1KDM1ACYP17A1CYP3A4CYP11B1
SCHEMBL9340840 0.69 TP53 (0.42) BACE1TP53PDK2ALDH1A1TDP1
SCHEMBL7072344 0.69 SLC18A3 (0.43) APPBACE1SIGMAR1KDM1ACYP17A1
SCHEMBL12291014 0.69 BACE1 (0.41) APPBACE1TP53KDM1AOPRM1
SCHEMBL1143677 0.69 CYP3A4 (0.46) APPBACE1SIGMAR1KDM1AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356915-A Antihypertensive and bronchodilator agents J. URIACH & CIA. S.A. (ES) 1994-10-18 US disclosed
EP-0600147-A1 Tetralones with pharmacological activity, compositions containing them and process for their preparation J. URIACH & CIA. S.A. (ES) 1994-06-08 EP disclosed