SCHEMBL9348407

SCHEMBL9348407

COc1cc(Br)c(COCc2ccccc2)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.48
TSHR P16473 1/20 0.46
MAOB P27338 1/20 0.44
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALOX5 P09917 1/20 0.41
ABCB1 P08183 2/20 0.40
CD274 Q9NZQ7 1/20 0.39
TAS2R14 Q9NYV8 1/20 0.39
PPARG P37231 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
ACHE P22303 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9352484 0.84 PTPN1 (0.47) PTPN1TSHRMAOBCA1CA2
SCHEMBL9349724 0.84 PTPN1 (0.47) PTPN1TSHRMAOBCA1CA2
SCHEMBL9352494 0.81 TSHR (0.44) TSHRCA1CA2TDP1ALOX5
SCHEMBL9348507 0.78 PTPN1 (0.45) PTPN1TDP1L3MBTL1TAS2R14HTR1A
SCHEMBL9349868 0.78 CRHR1 (0.35) PTPN1CA1CA2ALOX5ALDH1A1
SCHEMBL12772157 0.77 KMT2A (0.60) MAOBTDP1ABCB1PPARGALDH1A1
SCHEMBL4002789 0.76 ALDH1A1 (0.46) PTPN1CA1CA2ALDH1A1CYP1A2
SCHEMBL18029929 0.75 LTA4H (0.57) PTPN1TSHRMAOBCA1CA2
SCHEMBL9348530 0.75 MAOB (0.50) TSHRMAOBTDP1L3MBTL1ABCB1
SCHEMBL5956203 0.73 PTPN1 (0.58) PTPN1MAOBCA1CA2CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO claimed
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed