SCHEMBL9348779

SCHEMBL9348779

CC(C)(C)c1cc(-c2ncsn2)cc(C(C)(C)C)c1O

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
PTGS1 P23219 10/20 0.51
PTGS2 P35354 10/20 0.51
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2470646 0.75 CA2 (0.70) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL29090330 0.73 CA2 (0.59) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL803157 0.72 CA2 (1.00) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL2340718 0.69 CA2 (0.53) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL11868254 0.68 CA2 (0.57) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL10790942 0.68 CA2 (0.52) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL13722510 0.67 PTGS1 (0.73) CA1CA2PTGS1PTGS2CYP1A2
SCHEMBL9457150 0.67 SMPD3 (0.58) CA1CA2PTGS1PTGS2
SCHEMBL8766812 0.67 PTGS1 (0.58) CA1CA2PTGS1PTGS2
SCHEMBL9181713 0.66 CA1 (0.53) CA1CA2PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2270865-A None JP disclosed
US-5376670-A 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1994-12-27 US disclosed
US-5256680-A 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1993-10-26 US disclosed
US-5155122-A Cyclooxygenase, lipoxygenase inhibitors WARNER-LAMBERT COMPANY (US) 1992-10-13 US disclosed
JP-H02270865-A 3,5-DI-TERTIARY-BUTYL-4-HYDROXYPHENYL-1,3,4-THIADIAZOLE AND OXADIAZOLE, AND 3,5-DI-TERTIARY-BUTYL-4-HYDROXYPHENYL-1,2,4-THIADIAZOLE, OXADIAZOLE AND TRIAZOLE WARNER LAMBERT CO 1990-11-05 JP disclosed