SCHEMBL9350163

SCHEMBL9350163

Cc1csc2c(N)cccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
CYP3A4 P08684 4/20 0.42
TSHR P16473 3/20 0.42
TDP1 Q9NUW8 3/20 0.42
HSD17B10 Q99714 3/20 0.42
HPGD P15428 2/20 0.42
CD44 P16070 1/20 0.41
PIK3CA P42336 1/20 0.41
KDM4E B2RXH2 2/20 0.39
CYP2A6 P11509 3/20 0.37
CYP1A2 P05177 3/20 0.37
KEAP1 Q14145 1/20 0.37
NR4A2 P43354 1/20 0.34
PKM P14618 1/20 0.34
PARP1 P09874 2/20 0.34
CYP17A1 P05093 1/20 0.33
ELANE P08246 1/20 0.33
NSD2 O96028 2/20 0.32
MEN1 O00255 1/20 0.32
TDP2 O95551 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404365 0.80 CYP1A2 (0.48) ALDH1A1TSHRHSD17B10HPGDCYP2A6
SCHEMBL10338252 0.80 ALDH1A1 (0.48) ALDH1A1CYP3A4TSHRTDP1HSD17B10
SCHEMBL29908309 0.75 CYP2A6 (0.42) ALDH1A1CYP2A6CYP1A2NR4A2PARP1
SCHEMBL2090970 0.75 CYP2A6 (0.37) ALDH1A1CYP2A6CYP1A2CYP17A1
SCHEMBL30640459 0.75 ALDH1A1 (0.39) ALDH1A1CYP2A6CYP1A2CYP17A1
SCHEMBL10832904 0.75 TRPA1 (0.41) ALDH1A1TSHRTDP1HSD17B10HPGD
SCHEMBL2091920 0.75 ALDH1A1 (0.39) ALDH1A1CYP2A6CYP1A2CYP17A1
SCHEMBL787846 0.75 CYP2A6 (0.42) ALDH1A1CYP2A6CYP1A2NR4A2PARP1
SCHEMBL288465 0.75 ACHE (0.39) ALDH1A1TSHRCYP2A6CYP1A2CYP17A1
SCHEMBL4420462 0.74 CYP2A6 (0.41) CYP2A6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0340010-B1 Heterocyclic nitromethane derivatives ICI PLC (GB) 1994-08-24 EP disclosed
US-5102905-A For treating side effects of diabetes and galactosemia IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-04-07 US disclosed
EP-0340010-A2 Heterocyclic nitromethane derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-11-02 EP disclosed