SCHEMBL9352178

SCHEMBL9352178

Cn1c2ccccc2c(=O)c2c(O)cccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 1.00
MAPT P10636 1/20 1.00
CYP2C19 P33261 2/20 0.56
HSD17B10 Q99714 2/20 0.56
ALDH1A1 P00352 2/20 0.56
KDM4E B2RXH2 1/20 0.56
GLA P06280 1/20 0.56
GAA P10253 1/20 0.56
HPGD P15428 1/20 0.56
KDM1A O60341 1/20 0.52
GPR3 P46089 1/20 0.50
ATM Q13315 1/20 0.49
MAOA P21397 2/20 0.49
G6PD P11413 1/20 0.47
ERCC1 P07992 1/20 0.45
FEN1 P39748 1/20 0.45
ERCC4 Q92889 1/20 0.45
NTRK1 P04629 2/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2098721 0.85 MAPT (0.74) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL31265892 0.82 HTT (0.69) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL14802158 0.81 MAPT (0.68) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL10167907 0.79 HTT (0.66) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL10977307 0.79 HTT (0.66) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL382974 0.79 HTT (0.66) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL3875044 0.79 MAPT (0.63) HTTMAPTHSD17B10ALDH1A1KDM4E
SCHEMBL29466066 0.79 GPR3 (0.71) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL53107 0.79 GPR3 (0.71) HTTMAPTCYP2C19HSD17B10ALDH1A1
SCHEMBL21312375 0.79 GPR3 (0.71) HTTMAPTCYP2C19HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed