SCHEMBL9352575

SCHEMBL9352575

COc1cc(Nc2cc([N+](=O)[O-])ccc2C(=O)O)c(OC)c(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.56
AKR1C2 P52895 3/20 0.56
PKM P14618 2/20 0.52
CTSV O60911 1/20 0.50
CTSL P07711 1/20 0.50
KDM4E B2RXH2 1/20 0.49
POLB P06746 2/20 0.48
ANO1 Q5XXA6 1/20 0.48
ANO2 Q9NQ90 1/20 0.48
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
HTT P42858 3/20 0.48
MAPT P10636 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
GAA P10253 1/20 0.48
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
MPO P05164 1/20 0.47
LMNA P02545 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11235113 0.80 ALDH1A1 (0.58) PKMKDM4EMEN1KMT2AMAPT
SCHEMBL16737204 0.79 CDC25B (0.67) AKR1C3AKR1C2CTSVCTSLKDM4E
SCHEMBL16737123 0.77 ANO1 (0.58) AKR1C3AKR1C2CTSVCTSLPOLB
SCHEMBL380803 0.76 HTT (0.60) AKR1C3AKR1C2PKMCTSVCTSL
SCHEMBL22720115 0.75 MYC (0.65) AKR1C3AKR1C2CTSVCTSLMEN1
Hydrochloric Acid SCHEMBL6224359 0.75 HTT (0.58) AKR1C3AKR1C2PKMCTSVCTSL
Water SCHEMBL10360760 0.75 HTT (0.58) AKR1C3AKR1C2PKMCTSVCTSL
SCHEMBL16737120 0.74 ANO1 (0.84) AKR1C3AKR1C2CTSVCTSLPOLB
SCHEMBL16737205 0.74 ANO1 (0.62) AKR1C3AKR1C2PKMCTSVCTSL
SCHEMBL1671926 0.73 CTSV (0.60) PKMCTSVCTSLKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO claimed
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed