SCHEMBL9353040

SCHEMBL9353040

COc1ccc2c(C(C(=O)O)C(=O)O)cccc2c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
MTNR1A P48039 9/20 0.48
MTNR1B P49286 7/20 0.48
AKR1C3 P42330 6/20 0.48
AKR1C2 P52895 6/20 0.48
PTGS2 P35354 3/20 0.48
PTGS1 P23219 3/20 0.48
CYP1A2 P05177 2/20 0.48
CDC42 P60953 1/20 0.48
RAC1 P63000 1/20 0.48
TSHR P16473 1/20 0.48
SLC22A6 Q4U2R8 1/20 0.48
CYP2A6 P11509 1/20 0.44
AKR1C1 Q04828 1/20 0.44
HTR2C P28335 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7059358 0.87 PTGS2 (0.57) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2
SCHEMBL6280665 0.87 MTNR1A (0.48) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2
SCHEMBL7031139 0.87 PTGS2 (0.57) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2
Ammonia Solution, Strong SCHEMBL10891516 0.85 PTGS2 (0.56) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2
SCHEMBL27890994 0.85 PTGS2 (0.56) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2
SCHEMBL9483087 0.83 MTNR1A (0.47) KDM4EMTNR1AMTNR1BCYP1A2TSHR
SCHEMBL7379672 0.83 AKR1C3 (0.60) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2
SCHEMBL3929101 0.80 CYP2D6 (0.50) KDM4EMTNR1AMTNR1BCYP1A2CYP2A6
SCHEMBL3929104 0.80 CYP2D6 (0.50) KDM4EMTNR1AMTNR1BCYP1A2CYP2A6
SCHEMBL27581533 0.79 MTNR1A (0.46) KDM4EMTNR1AMTNR1BAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0461958-B1 2-(aminoalkyl)-5-(arylalkyl)1,3-dioxanderivatives their production and their use in therapeutics SYNTHELABO (FR) 1994-09-14 EP disclosed
EP-0461958-A1 2-(aminoalkyl)-5-(arylalkyl)1,3-dioxanderivatives their production and their use in therapeutics SYNTHELABO (FR) 1991-12-18 EP disclosed