SCHEMBL9353452

SCHEMBL9353452

CCCCCCCCOC(=O)CNC(=O)OCC#CI

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE P22303 12/20 0.46
NAAA Q02083 1/20 0.46
EPHX1 P07099 1/20 0.44
FAAH O00519 2/20 0.43
RAD52 P43351 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9353154 0.82 GAA (0.31)
SCHEMBL7565114 0.81 EPHX1 (0.56) ACHEEPHX1
SCHEMBL9189503 0.81 EPHX1 (0.56) ACHEEPHX1
SCHEMBL677759 0.81 EPHX1 (0.56) ACHEEPHX1
SCHEMBL677758 0.79 ACHE (0.59) ACHENAAAEPHX1
SCHEMBL6688663 0.79 ACHE (0.53) ACHEEPHX1
SCHEMBL9481159 0.79 GAA (0.58) FAAH
SCHEMBL6688659 0.77 ACHE (0.56) ACHEEPHX1
Iodocarb SCHEMBL114369 0.77 ACHE (0.59) ACHEEPHX1
SCHEMBL11308601 0.77 NAAA (0.47) ACHENAAAEPHX1FAAHRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490566-B1 Preparation and use of N-iodopropargyl oxycarbonyl amino acid esters and derivatives as antimicrobial agents ROHM & HAAS (US) 1994-10-12 EP claimed
US-5209930-A PREPARATION AND USE OF N-IODOPROPARGYL OXYCARBONYL AMINO ACID ESTERS AND DERIVATIVES AS ANTIMICROBIAL AGENTS ROHM AND HAAS COMPANY (US) 1993-05-11 US claimed
EP-0490566-A1 Preparation and use of N-iodopropargyl oxycarbonyl amino acid esters and derivatives as antimicrobial agents ROHM AND HAAS COMPANY (US) 1992-06-17 EP claimed
EP-0490566-B1 Preparation and use of N-iodopropargyl oxycarbonyl amino acid esters and derivatives as antimicrobial agents ROHM & HAAS (US) 1994-10-12 EP disclosed
US-5209930-A PREPARATION AND USE OF N-IODOPROPARGYL OXYCARBONYL AMINO ACID ESTERS AND DERIVATIVES AS ANTIMICROBIAL AGENTS ROHM AND HAAS COMPANY (US) 1993-05-11 US disclosed
EP-0490566-A1 Preparation and use of N-iodopropargyl oxycarbonyl amino acid esters and derivatives as antimicrobial agents ROHM AND HAAS COMPANY (US) 1992-06-17 EP disclosed