SCHEMBL9358367

SCHEMBL9358367

COc1cccc2c1C(C)(C)CCC2

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 1/20 0.44
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
KDM1A O60341 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ADRA2B P18089 1/20 0.39
PTGS1 P23219 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ADRA2A P08913 2/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
DRD1 P21728 1/20 0.37
DRD5 P21918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23023377 0.95 HTR5A (0.46) HTR5ADRD2DRD3ALDH1A1ADRA2B
SCHEMBL18053266 0.89 HTR5A (0.46) HTR5ADRD2DRD3ALDH1A1ADRA2B
SCHEMBL20445640 0.79 KDM1A (0.47) KDM1AALDH1A1TDP1MEN1KMT2A
SCHEMBL26889686 0.79 HTR5A (0.42) HTR5ADRD2DRD3ALDH1A1ADRA2B
SCHEMBL9457900 0.77 HTR5A (0.40) HTR5ADRD2DRD3MEN1KMT2A
SCHEMBL3908655 0.76 HTR5A (0.39) HTR5ADRD2DRD3MEN1KMT2A
SCHEMBL29823229 0.76 DRD2 (0.49) HTR5ADRD2DRD3ALDH1A1ADRA2B
SCHEMBL13999138 0.76 DRD2 (0.49) HTR5ADRD2DRD3ALDH1A1ADRA2B
SCHEMBL17014343 0.75 HTR5A (0.47) HTR5ADRD2DRD3ALDH1A1ADRA2B
SCHEMBL9358616 0.74 BCL2L1 (0.47) DRD2DRD3KDM1AALDH1A1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021032218-A1 HETEROCYCLIC THR-β RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREFOR 苏州闻天医药科技有限公司 2021-02-25 WO disclosed
EP-0418064-B1 Naphthalene and tetrahydronaphthalene gem-diphosphonate derivatives SYMPHAR SA (CH) 1994-12-14 EP disclosed
US-5204336-A Anticholestrol agents SYMPHAR S.A. (CH) 1993-04-20 US disclosed
EP-0418064-A2 Naphthalene and tetrahydronaphthalene gem-diphosphonate derivatives SYMPHAR S.A. (CH) 1991-03-20 EP disclosed