SCHEMBL9457900

SCHEMBL9457900

COc1cccc2c1C(CO)(CO)CCC2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 1/20 0.40
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
HTR7 P34969 1/20 0.35
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8139004 0.77 ALDH1A1 (0.44)
SCHEMBL3908655 0.77 HTR5A (0.39) HTR5ADRD2DRD3LMNASMN1; SMN2
SCHEMBL9358367 0.77 HTR5A (0.44) HTR5ADRD2DRD3LMNASMN1; SMN2
SCHEMBL26889686 0.74 HTR5A (0.42) HTR5ADRD2DRD3ADRA2A
SCHEMBL23023377 0.72 HTR5A (0.46) HTR5ADRD2DRD3LMNASMN1; SMN2
SCHEMBL13999138 0.71 DRD2 (0.49) HTR5ADRD2DRD3ADRA2A
SCHEMBL29823229 0.71 DRD2 (0.49) HTR5ADRD2DRD3ADRA2A
SCHEMBL17014343 0.70 HTR5A (0.47) HTR5ADRD2DRD3MEN1KMT2A
SCHEMBL13647144 0.70 IDO1 (0.41) HTR5ADRD2DRD3LMNASMN1; SMN2
SCHEMBL29598562 0.69 KDM1A (0.46) DRD2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5244888-A Hexahydroindenopyrroles and hexahydrobenzisoindoles ABBOTT LABORATORIES (US) 1993-09-14 US disclosed
US-5049564-A Hypotensive, 5-hydroxytryptamine ABBOTT LABORATORIES (US) 1991-09-17 US disclosed
EP-0422134-A1 5-HT SELECTIVE AGENTS. ABBOTT LAB (US) 1991-04-17 EP disclosed
WO-1990006927-A1 5-HT SELECTIVE AGENTS ABBOTT LABORATORIES (US) 1990-06-28 WO disclosed