SCHEMBL93596

SCHEMBL93596

CCCc1nc2c(n1Cc1ccc(-c3ccccc3-c3nnn[nH]3)cc1)CCCCC2=O

nearest known ligand 0.71

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 16/20 0.71
AGTR1 P30556 15/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9077559 0.86 AGTR2 (0.75) AGTR2AGTR1
Pratosartan SCHEMBL93595 0.86 AGTR1 (0.73) AGTR2AGTR1
SCHEMBL683741 0.85 AGTR1 (0.72) AGTR2AGTR1
SCHEMBL1652186 0.84 AGTR2 (0.90) AGTR2AGTR1
SCHEMBL9078950 0.83 AGTR2 (0.62) AGTR2AGTR1
SCHEMBL9007544 0.81 AGTR2 (0.49) AGTR2AGTR1
SCHEMBL7309330 0.81 AGTR1 (0.55) AGTR2AGTR1
SCHEMBL683401 0.81 AGTR1 (0.74) AGTR2AGTR1
SCHEMBL683452 0.80 AGTR1 (0.73) AGTR2AGTR1
SCHEMBL9844095 0.80 AGTR1 (0.51) AGTR2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2032 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-12016835-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2024-06-25 US claimed
US-20240173302-A1 TREATMENT OF INFLAMMATORY DISEASES DIMERIX BIOSCIENCE PTY LTD. (AU) 2024-05-30 US claimed
US-11931341-B2 Compositions and methods for the treatment and prevention of muscular dystrophy UNIVERSITY OF LOWA RESEARCH FOUNDATION (US) 2024-03-19 US claimed
EP-4313024-A1 TREATMENT OF INFLAMMATORY DISEASES Dimerix Bioscience Pty Ltd (AU) 2024-02-07 EP claimed
US-11851443-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-12-26 US claimed
US-20230285340-A1 NEPRILYSIN INHIBITORS THERAVANCE BIOPHARMA R&D IP LLC (US) 2023-09-14 US claimed
US-11718591-B2 Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2- methylpentanoic acid and uses thereof THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-08-08 US claimed
US-11634413-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-04-25 US claimed
WO-2022198264-A1 TREATMENT OF INFLAMMATORY DISEASES DIMERIX BIOSCIENCE PTY LTD (AU) 2022-09-29 WO claimed
WO-2005070463-A2 COMPOSITIONS COMPRISING (S)-AMLODIPINE MALATE AND AN ANGIOTENSIN RECEPTOR BLOCKER AND METHODS OF THEIR USE SEPRACOR, INC. (US) 2005-08-04 WO claimed
WO-2005070462-A2 COMPOSITIONS COMPRISING (S)-AMLODIPINE AND AN ANGIOTENSIN RECEPTOR BLOCKER AND METHODS OF THEIR USE SEPRACOR, INC. (US) 2005-08-04 WO claimed
US-20050143435-A1 Pharmaceutical compositions comprising a selective I1 imidazoline receptor agonist and an angiotensin II receptor blocker SOLVAY PHARMACEUTICALS GMBH (DE) 2005-06-30 US claimed
EP-1545540-A2 COMBINATION THERAPY USING A DUAL PPAR ALPHA/GAMMA AGONIST AND AN ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST Merck & Co., Inc. (US) 2005-06-29 EP claimed
WO-2005039639-A2 PHARMACEUTICAL COMPOSITION COMPRISING A SELECTIVE I1 IMIDAZOLINE RECEPTOR AGONIST AND AN ANGIOTENSIN II RECEPTOR BLOCKER SOLVAY PHARMACEUTICALS GMBH (DE) 2005-05-06 WO claimed
WO-2005039638-A2 THERAPEUTIC AGENT FOR HEART FAILURE COMPRISING AN ANGIOTENSIN II RECEPTOR ANTAGONIST AND A MATRIX METALLOPROTEINASE INHIBITOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-05-06 WO claimed
WO-2005000217-A2 COMBINATION THERAPY FOR THE TREATMENT OF DYSLIPIDEMIA MERCK & CO., INC. (US) 2005-01-06 WO claimed
WO-2004110375-A2 COMBINATION THERAPY FOR THE TREATMENT OF DIABETES MERCK & CO., INC. (US) 2004-12-23 WO claimed
WO-2004089416-A2 COMBINATION OF AN 11BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITOR AND AN ANTIHYPERTENSIVE AGENT NOVO NORDISK A/S (DK) 2004-10-21 WO claimed
WO-2004017896-A2 COMBINATION THERAPY USING A DUAL PPAR ALPHA/GAMMA AGONIST AND AN ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST MERCK & CO., INC. (US) 2004-03-04 WO claimed