SCHEMBL936280

SCHEMBL936280

CCC(C#N)NC(=O)c1cc(F)cc(-c2cc(-c3ccc(N4CCN(C)CC4)c(Cl)c3)[nH]n2)c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 15/20 0.51
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MELK Q14680 1/20 0.36
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36
WDR5 P61964 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6924025 0.91 PRKD1 (0.55) PRKD1ALDH1A1L3MBTL1MELKWDR5
SCHEMBL6922437 0.87 PRKD1 (0.67) PRKD1ALDH1A1L3MBTL1MELKHTR1A
SCHEMBL1056933 0.80 PRKD1 (0.68) PRKD1
SCHEMBL936747 0.80 PRKD1 (0.68) PRKD1
SCHEMBL936380 0.78 PRKD1 (0.76) PRKD1MELK
SCHEMBL6922426 0.77 PRKD1 (0.82) PRKD1MELKWDR5
SCHEMBL936340 0.77 PRKD1 (0.83) PRKD1MELK
SCHEMBL6924016 0.74 PRKD1 (0.67) PRKD1MELK
SCHEMBL960572 0.72 PRKD1 (0.64) PRKD1MELKWDR5
SCHEMBL1083601 0.71 PRKD1 (0.81) PRKD1MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009484-A1 ARYLPYRAZOLES AND ARYLISOXAZOLES AND THEIR USE AS PKD MODULATORS NOVARTIS AG (CH) 2011-01-27 WO disclosed
WO-2011009484-A1 ARYLPYRAZOLES AND ARYLISOXAZOLES AND THEIR USE AS PKD MODULATORS NOVARTIS AG (CH) 2011-01-27 WO disclosed