SCHEMBL936340

SCHEMBL936340

CN1CCN(c2ccc(-c3cc(-c4cccc(C(=O)NCC#N)c4)n[nH]3)cc2Cl)CC1

nearest known ligand 0.83

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 16/20 0.83
PAK1 Q13153 1/20 0.53
MELK Q14680 1/20 0.44
FLT3 P36888 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6922437 0.89 PRKD1 (0.67) PRKD1PAK1MELK
SCHEMBL1056933 0.86 PRKD1 (0.68) PRKD1
SCHEMBL936747 0.86 PRKD1 (0.68) PRKD1
SCHEMBL6922426 0.85 PRKD1 (0.82) PRKD1MELK
SCHEMBL6924254 0.85 PRKD1 (0.78) PRKD1PAK1MELKFLT3
SCHEMBL960572 0.84 PRKD1 (0.64) PRKD1PAK1MELKFLT3BCHE
SCHEMBL6923773 0.83 PRKD1 (0.78) PRKD1PAK1
SCHEMBL6924016 0.82 PRKD1 (0.67) PRKD1MELKFLT3
SCHEMBL936181 0.80 PRKD1 (1.00) PRKD1MELKFLT3
SCHEMBL936280 0.77 PRKD1 (0.51) PRKD1MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009484-A1 ARYLPYRAZOLES AND ARYLISOXAZOLES AND THEIR USE AS PKD MODULATORS NOVARTIS AG (CH) 2011-01-27 WO disclosed