SCHEMBL9364248

SCHEMBL9364248

COCCOC(=O)OC1=C(C)N(C)C(C)=C(OC(=O)OC)C1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GPBAR1 Q8TDU6 1/20 0.39
HTT P42858 2/20 0.38
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
LMNA P02545 1/20 0.37
RECQL P46063 1/20 0.37
KMT2A Q03164 1/20 0.36
HPGD P15428 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CACNA1F O60840 1/20 0.36
CACNA1D Q01668 1/20 0.36
CACNA1S Q13698 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9364254 0.92 HSP90AA1 (0.40) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9364015 0.92 HSP90AA1 (0.42) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL8984936 0.90 HSP90AA1 (0.46) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9364528 0.85 NPSR1 (0.45) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9363808 0.84 HSP90AA1 (0.42) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9220730 0.82 APOBEC3A (0.36) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9364057 0.82 HSP90AA1 (0.41) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9364594 0.81 KDM4E (0.42) HSP90AA1HSP90AB1KDM4EALDH1A1GAA
SCHEMBL9215408 0.80 KDM4E (0.37) KDM4EALDH1A1GAAPOLBTDP1
SCHEMBL7428174 0.80 HSP90AA1 (0.43) HSP90AA1HSP90AB1KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP claimed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP claimed
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP disclosed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP disclosed