SCHEMBL9364645

SCHEMBL9364645

CCOC(=O)C(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 4/20 0.68
ALDH1A1 P00352 4/20 0.57
MAPT P10636 2/20 0.56
NPSR1 Q6W5P4 1/20 0.49
LMNA P02545 1/20 0.49
THRA P10827 1/20 0.48
THRB P10828 1/20 0.48
P2RX1 P51575 2/20 0.48
ACP1 P24666 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
HPGD P15428 1/20 0.46
TMPRSS4 Q9NRS4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23167797 0.93 GPR35 (0.63) GPR35ALDH1A1MAPTNPSR1LMNA
SCHEMBL596433 0.85 ALDH1A1 (0.60) GPR35ALDH1A1MAPTNPSR1LMNA
SCHEMBL24969427 0.84 MAPT (0.69) GPR35ALDH1A1MAPTNPSR1HPGD
SCHEMBL11400761 0.81 GPR35 (1.00) GPR35ALDH1A1MAPTHPGD
SCHEMBL7692960 0.79 GPR35 (0.74) GPR35MAPTLMNAP2RX1ACP1
SCHEMBL25780344 0.79 GPR35 (0.57) GPR35ALDH1A1NPSR1THRBP2RX1
SCHEMBL9364641 0.79 GPR35 (0.59) GPR35ALDH1A1MAPTLMNAP2RX1
SCHEMBL5973284 0.78 GPR35 (0.67) GPR35ALDH1A1MAPTNPSR1LMNA
SCHEMBL25247718 0.77 GPR35 (0.54) GPR35ALDH1A1MAPTNPSR1HPGD
SCHEMBL17209749 0.77 GAA (0.49) GPR35ALDH1A1MAPTNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377112-B1 Quinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-08-24 EP disclosed
US-5061706-A 2,3-QUINOXALINEDIONES FOR USE AS NEUROLEPTICS NOVO NORDISK A/S (DK) 1991-10-29 US disclosed
EP-0377112-A1 Quinoxaline compounds and their preparation and use NOVO NORDISK A/S (DK) 1990-07-11 EP disclosed