SCHEMBL9367707

SCHEMBL9367707

C1=C(c2ccccc2)CCC(CN2CCN(c3ccccn3)CC2)C1

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.51
DRD4 P21917 2/20 0.51
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
DRD3 P35462 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9370055 0.89 DRD2 (0.49) DRD2DRD4HTR2AHTR2C
SCHEMBL7783724 0.89 DRD2 (0.54) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL9371451 0.88 DRD2 (0.56) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL9367241 0.85 DRD2 (0.45) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL7783722 0.82 DRD2 (0.58) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL7792010 0.82 DRD2 (0.58) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL13648727 0.80 DRD2 (0.62) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL9367644 0.80 DRD3 (0.55) DRD2DRD4HTR2AHTR2CDRD3
SCHEMBL9367787 0.79
SCHEMBL9367275 0.78 DRD2 (0.55) DRD2DRD4HTR2AHTR2CDRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP claimed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP disclosed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4975445-A Antidepressants WARNER-LAMBERT COMPANY (US) 1990-12-04 US disclosed