SCHEMBL9367275

SCHEMBL9367275

C1=C(c2ccccn2)CCC(CCN2CCN(c3ccccn3)CC2)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.55
DRD3 P35462 4/20 0.55
HTR1A P08908 3/20 0.52
DRD4 P21917 3/20 0.51
HTR2C P28335 3/20 0.51
HTR2A P28223 2/20 0.51
HTR7 P34969 2/20 0.51
SLC6A4 P31645 1/20 0.48
SIGMAR1 Q99720 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9371451 0.90 DRD2 (0.56) DRD2DRD3HTR1ADRD4HTR2C
SCHEMBL9370055 0.89 DRD2 (0.49) DRD2DRD4HTR2CHTR2A
SCHEMBL9367644 0.86 DRD3 (0.55) DRD2DRD3HTR1ADRD4HTR2C
SCHEMBL9368439 0.84 DRD2 (0.54) DRD2DRD3HTR1ADRD4HTR2C
SCHEMBL9367665 0.84 HTR2C (0.53) DRD2DRD3HTR1ADRD4HTR2C
SCHEMBL8470779 0.79 DRD2 (0.65) DRD2DRD3HTR1ADRD4HTR2C
SCHEMBL9367707 0.78 DRD2 (0.51) DRD2DRD3DRD4HTR2CHTR2A
SCHEMBL2021022 0.78
SCHEMBL9195812 0.76 DRD2 (0.61) DRD2DRD3HTR1ADRD4HTR2C
SCHEMBL3849926 0.75 DRD2 (0.70) DRD2DRD3HTR1ADRD4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP claimed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP disclosed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4975445-A Antidepressants WARNER-LAMBERT COMPANY (US) 1990-12-04 US disclosed