SCHEMBL9367644

SCHEMBL9367644

Fc1ccc(C2=CCC(CCN3CCN(c4ccccn4)CC3)CC2)cc1

nearest known ligand 0.84

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 8/20 0.55
DRD2 P14416 7/20 0.55
HTR1A P08908 6/20 0.55
HTR2A P28223 5/20 0.55
HTR7 P34969 5/20 0.55
DRD4 P21917 3/20 0.55
SIGMAR1 Q99720 3/20 0.55
SLC6A4 P31645 2/20 0.55
HTR2C P28335 1/20 0.55
ADRA2C P18825 3/20 0.53
DRD1 P21728 3/20 0.53
DRD5 P21918 3/20 0.53
HRH1 P35367 3/20 0.53
SLC6A2 P23975 1/20 0.51
SLC6A3 Q01959 1/20 0.51
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9371451 0.91 DRD2 (0.56) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9367275 0.86 DRD2 (0.55) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9368439 0.82 DRD2 (0.54) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9367665 0.82 HTR2C (0.53) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9367707 0.80 DRD2 (0.51) DRD3DRD2HTR2ADRD4HTR2C
SCHEMBL8470779 0.76 DRD2 (0.65) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL7788928 0.76 MAPT (0.52) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9195812 0.76 DRD2 (0.61) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9200413 0.75 DRD2 (0.55) DRD3DRD2HTR1AHTR2AHTR7
SCHEMBL9370055 0.75 DRD2 (0.49) DRD2HTR2ADRD4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP claimed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP disclosed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4975445-A Antidepressants WARNER-LAMBERT COMPANY (US) 1990-12-04 US disclosed