SCHEMBL9370802

SCHEMBL9370802

CCOC(=O)c1cc(CC)cnc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
ALDH1A1 P00352 3/20 0.48
TSHR P16473 2/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.46
CYP4F2 P78329 1/20 0.45
CYP4A11 Q02928 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
RAB9A P51151 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HPGD P15428 2/20 0.44
HSP90AA1 P07900 2/20 0.44
GAA P10253 2/20 0.44
MAPK1 P28482 1/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28166126 0.87 KDM4E (0.46) KDM4EALDH1A1TSHRALOX15HSD17B10
SCHEMBL6559833 0.85 TSHR (0.46) KDM4EALDH1A1TSHRCYP4F2CYP4A11
SCHEMBL29897883 0.85 TSHR (0.46) KDM4EALDH1A1TSHRCYP4F2CYP4A11
SCHEMBL25255731 0.85 KDM4E (0.49) KDM4EALDH1A1TSHRALOX15HSD17B10
SCHEMBL29501650 0.85 KDM4E (0.49) KDM4EALDH1A1TSHRALOX15HSD17B10
SCHEMBL612735 0.84 KDM4E (0.51) KDM4EALDH1A1TSHRALOX15HSD17B10
SCHEMBL8627488 0.83 CYP4F2 (0.50) KDM4EALDH1A1TSHRCYP4F2CYP4A11
SCHEMBL277286 0.83 CYP2C9 (0.54) KDM4EALDH1A1TSHRALOX15HSD17B10
SCHEMBL12458000 0.83 CA12 (0.56) KDM4EALDH1A1TSHRALOX15HSD17B10
SCHEMBL9370371 0.82 GABRP (0.46) KDM4EALDH1A1TSHRALOX15MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220518-B1 PREPARATION OF SUBSTITUTED AND DISUBSTITUTED PYRIDINE-2,3-DICARBOXYLATE ESTERS AMERICAN CYANAMID COMPANY (US) 1991-02-06 EP claimed
US-4723011-A ALPHA-HALO-BETA-KETOESTERS, ALPHA, BETA UNSATURATED KETONE OR ALDEHYDE, AMMONIUM SALT AMERICAN CYANAMID COMPANY (US) 1988-02-02 US claimed
EP-0220518-A2 Preparation of substituted and disubstituted pyridine-2,3-dicarboxylate esters AMERICAN CYANAMID COMPANY (US) 1987-05-06 EP claimed
EP-0388620-B1 Process for the preparation of o-carboxypyridyl- and o-carboxyquinolylimidazolinones AMERICAN CYANAMID CO (US) 1994-11-02 EP disclosed
EP-0220518-B1 PREPARATION OF SUBSTITUTED AND DISUBSTITUTED PYRIDINE-2,3-DICARBOXYLATE ESTERS AMERICAN CYANAMID COMPANY (US) 1991-02-06 EP disclosed
EP-0388620-A1 Process for the preparation of o-carboxypyridyl- and o-carboxyquinolylimidazolinones AMERICAN CYANAMID COMPANY (US) 1990-09-26 EP disclosed
US-4925944-A CONDENSATION AND CYCLIZATION IN AROMATIC SOLVENT AND SULFUR; ONE STEP; HERBICIDES AMERICAN CYANAMID COMPANY (US) 1990-05-15 US disclosed
US-4723011-A ALPHA-HALO-BETA-KETOESTERS, ALPHA, BETA UNSATURATED KETONE OR ALDEHYDE, AMMONIUM SALT AMERICAN CYANAMID COMPANY (US) 1988-02-02 US disclosed
EP-0220518-A2 Preparation of substituted and disubstituted pyridine-2,3-dicarboxylate esters AMERICAN CYANAMID COMPANY (US) 1987-05-06 EP disclosed