SCHEMBL9370896

SCHEMBL9370896

Fc1ccc(-c2csc(NC(=S)N3CCN(C(c4ccc(F)cc4)c4ccc(F)cc4)CC3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.50
MEN1 O00255 6/20 0.50
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 4/20 0.45
MAOA P21397 3/20 0.44
MAOB P27338 3/20 0.44
MMP2 P08253 1/20 0.44
MMP8 P22894 1/20 0.44
MAPK1 P28482 2/20 0.44
POLB P06746 1/20 0.43
PRKACA P17612 1/20 0.43
ROCK1 Q13464 1/20 0.43
ALOX5 P09917 2/20 0.43
NR2F2 P24468 1/20 0.43
CDC25A P30304 1/20 0.43
CDC25B P30305 1/20 0.43
CDC25C P30307 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9371102 0.95 KMT2A (0.46) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9370694 0.95 KMT2A (0.48) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9370254 0.95 KMT2A (0.53) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9371270 0.92 KCNQ1 (0.49) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9370805 0.92 KDM4E (0.48) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9370589 0.89 KMT2A (0.50) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9370671 0.87 ROCK1 (0.55) KMT2AMEN1LMNAMMP2MMP8
SCHEMBL9375951 0.87 ALDH1A1 (0.54) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9376939 0.85 FAAH (0.43) KMT2AMEN1MAPTSMN1; SMN2LMNA
SCHEMBL9374499 0.84 ALDH1A1 (0.50) KMT2AMEN1MAPTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0589985-A1 2-AMINO-4-ARYL-THIAZOLES WITH ANTIASTHMATIC AND ANTI-INFLAMMATORY ACTIVITIES ON THE RESPIRATORY TRACT BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1994-04-06 EP disclosed
WO-1993000342-A1 2-AMINO-4-ARYL-THIAZOLES WITH ANTIASTHMATIC AND ANTI-INFLAMMATORY ACTIVITIES ON THE RESPIRATORY TRACT BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-01-07 WO disclosed
EP-0519449-A1 2-Amino-4-aryl thiazoles with antiasthmatic and antiinflammatory activities on the respiratory tract BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-12-23 EP disclosed