SCHEMBL9370964

SCHEMBL9370964

CS(=O)(=O)Nc1ccc2[nH]cc(CCC(=O)O)c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.64
HPGD P15428 2/20 0.59
CYP2C19 P33261 2/20 0.59
HTR6 P50406 6/20 0.49
HTR1A P08908 3/20 0.46
HTR1D P28221 2/20 0.46
CYP1A2 P05177 2/20 0.46
NQO2 P16083 1/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MPO P05164 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350200 0.89 HPGD (0.57) SPRHPGDCYP2C19HTR6CYP1A2
SCHEMBL14487470 0.87 SPR (0.60) SPRHPGDCYP2C19HTR6HTR1A
SCHEMBL9371511 0.84 SPR (0.62) SPRHPGDCYP2C19HTR6HTR1A
SCHEMBL2538876 0.83 SPR (0.61) SPRHPGDCYP2C19HTR6HTR1A
SCHEMBL14555323 0.83 SPR (0.60) SPRHPGDCYP2C19HTR6HTR1A
SCHEMBL12352688 0.82 SPR (0.67) SPRHPGDCYP2C19HTR6HTR1A
SCHEMBL21247057 0.82 HPGD (0.61) SPRHPGDCYP2C19HTR1AHTR1D
SCHEMBL8544819 0.82 HTR6 (0.59) HPGDCYP2C19HTR6MAPT
SCHEMBL4159606 0.81 SPR (0.46) SPRHPGDCYP2C19HTR6HTR1A
SCHEMBL14487812 0.80 SPR (0.64) SPRHPGDHTR6HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464558-B1 Antimigraine alkoxypyrimidine derivatives BRISTOL MYERS SQUIBB CO (US) 1994-12-28 EP disclosed
EP-0464558-A1 Antimigraine alkoxypyrimidine derivatives Bristol-Myers Squibb Company (US) 1992-01-08 EP disclosed